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抑制剂描述: 产品名称:Talmapimod (SCIO-469) 产品别名:见爱必信官网 英文别名:Talmapimod (SCIO-469) 靶点:p38 MAPK CAS:309913-83-5 纯度:98% 外观:见爱必信官网 保存方法:Store at -20°C 描述: Talmapimod (SCIO-469) is a selective ATP-competitive p38 inhibitor with IC50 of 9 nM for p38α.
Talmapimod (SCIO-469)decreased constitutive p38α MAPK phosphorylation of both 5T2MM and 5T33MM cells. Talmapimod (SCIO-469) also inhibits secretion and expression of the osteoclast-activating factors IL-11, receptor activator of NF-κB ligand, and macrophage inflammatory protein 1α, and prevents human osteoclast activationIn. It can also inhibit multiple myeloma growth and prevents bone disease in the 5T2MM and 5T33MM models.
Targeting p38α MAPK with Talmapimod (SCIO-469) decreases myeloma burden in addition to preventing the development of myeloma bone disease.
溶解性:Soluble in DMSO 体外研究: 体内研究:
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爱必信(上海)生物科技有限公司
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2010-12-13
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爱必信(上海) 生物科技有限公司
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