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一键询价MKN1 人胃癌细胞 QCH812
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Phoenix-AMPHO 人肾上皮细胞 QCH813
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SNU638 人胃癌细胞 QCH815
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NCI-H2073 人非小细胞肺癌细胞 QCH816
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HAL01 人急性淋巴细胞白血病细胞 QCH817
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TMD8 人弥漫性大B细胞淋巴瘤 QCH818
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SNU484 人胃癌细胞 QCH819
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JHH2 人肝癌细胞 QCH820
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LK2 人肺腺癌细胞 QCH821
钦诚生物 | 一周
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抑制剂描述: 产品名称:SUN 1334H 产品别名:见爱必信官网 英文别名:SUN 1334H 靶点:H1 receptor CAS:607736-84-5 纯度: 外观:见爱必信官网 保存方法:store at -20℃ for one year(Powder) 描述:SUN 1334H is a potent, orally active, highly selective H1 receptor antagonist, with Ki of 9.7 nM. 溶解性:DMSO* 体外研究: SUN-1334H causes potent inhibition of histamine induced contractions of isolated guinea-pig ileum with an IC50 (half the maximal inhibitory concentration) of 0.198 μM. In CHO-K1/hERG cells, SUN-1334H does not modulate hERG K+-currents at concentrations as high as 100 μM. SUN-1334H, cetirizine and hydroxyzine cause comparable inhibition of NLF leukocytes, IL-4 and total protein concentrations. 体内研究:SUN-1334H causes potent inhibition of histamine induced contractions of isolated guinea-pig ileum with an IC50 (half the maximal inhibitory concentration) of 0.198 μM. In CHO-K1/hERG cells, SUN-1334H does not modulate hERG K+-currents at concentrations as high as 100 μM. SUN-1334H, cetirizine and hydroxyzine cause comparable inhibition of NLF leukocytes, IL-4 and total protein concentrations.
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