Aminoglycoside derivatives 氨基糖苷类衍生物

规格: 5 mg, 25 mg, 100 mg, 1 g, 5 g

EOT-AMG001

氨基糖苷 平台1
Aminoglycoside platform 1

R1=H
R2=H
R1=PMB* with:
R2=(CH2)6Br or
(CH2)6N3 or
(CH2)6NH2 or
(CH2)6NHC(O)(CH2)2COOH
*PMB=para-methoxybenzyl, Tr=Trityl

EOT-AMG002

氨基糖苷 平台2
Aminoglycoside platform 2

R2=H: neamine
R2=(CH2)nBr or
(CH2)nN3 or
(CH2)nNH2 or
(CH2)6NHC(O)(CH2)2COOH or
(CH2)n-CH3
(n≥ 6)

EOT-AMG003

氨基糖苷 平台3
Aminoglycoside platform 3

R1=PMB with:
R2=H or
(CH2)nBr or
(CH2)nN3 or
(CH2)nNH2 or
(CH2)nNHC(O)(CH2)2COOH
(n≥ 6)
*PMB=para-methoxybenzyl, Tr=Trityl

EOT-AMG004

氨基糖苷 平台4
Aminoglycoside platform 4

R2=(CH2)nBr or
(CH2)nN3 or
(CH2)nNH2 or
(CH2)nNHC(O)(CH2)2COOH or
(CH2)n-CH3
(n≥ 4)